D-773

Determination of Mogroside V by HPLC-UV

Section D — Laboratory Operations and Specifications Revision 22 7 pages

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1.0 Purpose 
 
 This document describes the analytical procedure for the determination of mogroside V in raw
 materials and finished products. 
 
 2.0 Scope 
 
 This procedure applies to the identification and quantification of mogroside V in raw materials
 and finished products. This method was validated under Protocol MV-LAB-19-016.
 
 3.0 Responsibility 
 
 3.1 ‘It is the responsibility of QC and Analytical chemists who have verified their ability to
 
 execute this procedure to follow this procedure. 
 
 3.2 It is the responsibility of QC Laboratory Management to implement this procedure and
 to ensure that the procedure is being followed. 
 
 3.3. ‘It is the responsibility of QC Laboratory Management and/or Analytical Development
 to keep this procedure aligned with current laboratory practices. 
 
 4.0 Definitions 
 
 4.1 QC — Quality Control 
 
 4.2. AD-— Analytical Development 
 
 4.3 MGV- Mogroside V 
 
 4.4 ACN — Acetonitrile 
 
 
 

[SOP 

 Standard Operating Procedure SOPNo | Rev 
 Determination of Mogroside V by HPLC/UV D-773 22 eget 
 
 4.5 MeOH — Methanol 
 
 4.6 HPLC — High Performance Liquid Chromatography 
 
 5.0 References 
 
 5.1 MV-LAB-19-016, Protocol, Determination of Mogroside V using HPLC with UV/Vis
 
 Detection 
 
 5.2. RPT-23-0058, Report, Change of Mobile Phase for D-773 
 
 6.0 Supplies 
 
 6.1 Chemicals — All reagents are HPLC grade or better 
 
 6.1.1 ACN 
 
 6.1.2 MeOH 
 
 6.1.3 MGV Reference Standard 
 
 6.2 Supplies and Glassware 
 
 6.2.1 HPLC vials, 12mm X 32mm with screw cap enclosures w/ septa 
 
 6.2.2 Volumetric glassware and/or adjustable pipettes and tips 
 
 6.2.3 Weigh paper or funnels 
 
 6.2.4 1.5mL or 2.0mL micro centrifuge tubes 
 
 6.3 Equipment 
 
 6.3.1 Suitable gradient HPLC system consisting of a pump, autosampler, column oven
 and UV detector with a chromatographic data handling system 
 
 6.3.2 Analytical Balance 
 
 
 

[SOP 

 Standard Operating Procedure SOP No Rev 
 Determination of Mogroside V by HPLC/UV D-773 Page 3 of 7 
 
 6.3.3 Sonicator bath 
 
 6.3.4 Centrifuge 
 
 7.0 Procedure 
 
 Tel Mobile Phase Preparation 
 
 7.1.1 Mobile Phase 
 
 7.1.1.1 Combine 700 mL of ACN with 300 mL of water. 
 
 7.1.2 Diluent 
 
 7.1.2.1 MeOH 
 
 7.1.3 May be scaled as necessary 
 
 7.2. Standard Prep 
 
 7.2.1 Accurately weigh and transfer about 22 mg of MGV reference standard into a
 
 100-mL volumetric flask. 
 
 7.2.2 Dissolve in and dilute to volume with Diluent. 
 
 7.3. Sample Preparation 
 
 7.3.1 Specific sample testing details are provided in each products profile. If a
 
 specific testing details section is not available, then follow preparation
 procedure as described below, maintaining concentration within the linear range
 
 listed below. 
 
 7.3.2 The validated range for the analytical method is 0.06 — 0.29 mg/mL.
 
 7.3.3 For raw materials: weigh no less than 25 mg into a suitably sized volumetric
 flask of no less than 25 mL volume to generate an analyte concentration that is
 
 
 

[SOP 

 Standard Operating Procedure SOP No | Rev 
 Determination of Mogroside V by HPLC/UV D-773 2: || Rae OED 
 
 within the validated linearity range. Fill the flask to about 90% of the calculated
 
 volume with Diluent and sonicate for 10 minutes. Equilibrate to room
 
 temperature, and bring up to volume with Diluent. 
 
 7.3.4 For solid and liquid dose finished products: Combine and homogenize no less
 
 than ten dosage units. Based on the label claim and fill weight (capsules),
 serving size (powders and liquids) or tablet weight per dose, weigh no less than
 
 100 mg of the pooled dosages into a suitably sized volumetric flask of no less
 
 than 25 mL to generate an analyte concentration that is within the validated
 linear range. Fill the flask to about 90% of the calculated volume with Diluent
 
 and sonicate for 10 minutes. Equilibrate to room temperature, and bring up to
 volume with Diluent. 
 
 7.3.5 For chewable gels (gummies), homogenize at least 10 dosage units according to
 the procedure outlined in D-793 Cryogenic Grinding of Chewable Gels. Quickly
 
 weigh no less than 400 mg of the pooled and homogenized dosages into a
 
 suitably sized beaker. Add a volume of Diluent equivalent to 50% of the desired
 flask volume, cover the beaker opening, and sonicate for 10 minutes or until
 
 dissolved. Transfer the solution to a volumetric flask of size suitable to generate
 an analyte concentration that is within the validated linear range. Use several
 
 small portions of Diluent to rinse any remaining residue from the beaker into the
 
 volumetric flask ensuring complete transfer, and dilute to volume using Diluent.
 
 7.3.6 To manage large volumes, the sample can be initially dissolved in a smaller
 
 volume and a portion further diluted using Diluent to bring the analyte
 concentration into the linear range. Dilutions can be made using volumetric
 
 glassware and/or adjustable pipettes. Dilutions can be prepared in HPLC vials.
 
 7.3.7. Centrifuge an aliquot of the final sample at 10,000 rpm for 5 min to remove
 
 particulates. Alternatively, the sample may be filtered through a 0.45 um
 membrane discarding the first 3 — 4 mL before collecting a portion for analysis.
 
 
 

[SOP 

 Standard Operating Procedure SOP No | Rev 
 Determination of Mogroside V by HPLC/UV D-773 2 -|-RARE St 
 
 7.4 HPLC Parameters 
 
 7.4.1 Column: Hypersil Gold Amino Column 5pm x 4.6mm x 250mm 
 
 7.4.2 Column Temperature: Not controlled 
 
 7.4.3 Flow rate: 1.0 mL/min 
 
 7.4.4 Wavelength: 210 nm 
 
 7.4.5 Injection Volume: 10 pL 
 
 7.4.6 Run Time: 15 minutes 
 
 7.4.7 Recommended 3-D Spectral Range (for Identification): 200 nm - 400 nm
 
 7.5 Recommended Sequence 
 
 7.5.1. Make at least 2 injections of the diluent. 
 
 7.5.2 Make five (5) injections of Standard Solution. 
 
 7.5.3 Make a single injection of each Sample Preparation. 
 
 7.5.4 Make a single injection of the Standard Solution after every ten (10) sample
 
 injections or at the end of a run. 
 
 7.6 System Suitability Requirements 
 
 7.6.1 The %RSD of the first five (5) standard injections is NMT 3.0%.
 
 7.6.2 The %RSD of all standard injections is NMT 3%. 
 
 7.6.3 If present, any interference in the diluent should be subtracted out of the sample
 
 and standard peak areas. 
 
 7.7. Example calculations for determining finished product % label or raw material % purity
 
 
 

[SOP 

 Standard Operating Procedure SOP No | Rev 
 Determination of Mogroside V by HPLC/UV D-773 2. Rage G07 
 
 7.7.1 % MagrosidV e= Ruy WitaXP y S x Yet x 100 
 Ry Woe SA” LA 
 
 R., Sample peak area 
 
 R, Mean standard peak area 
 
 Wt,,, Weight of the reference standard in mg 
 
 Vs Volume of the standard preparation accounting for dilutions in mL
 
 P Purity of the reference standard in decimal format 
 
 SA Sample amount in mg 
 
 Woess Volume of the sample preparation accounting for dilutions in mL
 
 SS Serving size: Average weight of ten dosage units in mg for tablets,
 
 capsules, and gummies; weight of a single serving from the theoretical
 
 formula in mg for liquids and powders, or 1 for raw materials.
 
 LA Label amount in mg of mogroside V (use 1 for raw materials)
 
 7.8 Column Wash and Storage 
 
 7.8.1 Store the column in 100% ACN. 
 
 8.0 Chromatograms 
 
 8.1 Typical Diluent Chromatogram 
 
 DILUENT 
 64 
 2oO 
 54 
 44 
 34 
 > 3] 
 - 4 
 04 —_—~—— 
 “14 
 -24 
 -34 \ 
 44 \ 
 Hl 2 3 4 5 6 7 8 9 10.11 12 #13 «14 ~©«15 
 Time [min] 
 

[SOP 

 Standard Operating Procedure SOP No | Rev 
 Determination of Mogroside V by HPLC/UV D-773 2... Rage dot? 
 
 8.2 Typical Working Standard Chromatogram 
 
 SS 22AS021 STD 
 18; - 
 zB 
 16; 
 144 5, 
 124 FS 
 10; os 
 > 5 Ps 
 6 to) 
 44 2 = = 
 24 “ = 3 
 of _ bd 
 -2+ 
 44 
 -64 : ; . . ; . : ; : o ; : , : a 
 1 2 3 4 5 6 7 8 9 10 14 12 13 14 15 
 Time [min] 
 8.3. Typical Sample Chromatogram 
 RS50069 
 184 a ‘ 
 16+ i) 3 
 144 & 
 12+ = 
 10+ 
 2 84 
 @ 
 “ s 8 fe 
 -24 
 1 2 3 4 5 6 7 8 9 0 1 12 «2413 «14 © 15 
 Time (min] 
 
 9.0 Revision History 

| Rev | Date | Description of Changes | CCR # | By |
|-----|----------|------------------------|-------|----|
| 0 | 06/26/19 | New N/A S. Sassman | - | - |
| 1 | 06/22/22 | Updated logo and format. CC- Change mobile phase as discussed in RPT-23-0058, update | 22-0291 | K. Burris |
| 2 | 10/20/23 | example chromatograms, update sample prep section for CC- consistency with current methods, change column storage to be more appropriate for amino column. | 23-0522 | §. Sassman |